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Home - Products - GPCR/G Protein - Cannabinoid Receptor - Org 27569

Org 27569

CAS No. 868273-06-7

Org 27569 ( Org-27569;Org27569 )

Catalog No. M16306 CAS No. 868273-06-7

Org 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 28 In Stock
5MG 43 In Stock
10MG 73 In Stock
25MG 143 In Stock
50MG 267 In Stock
100MG 399 In Stock
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Biological Information

  • Product Name
    Org 27569
  • Note
    Research use only, not for human use.
  • Brief Description
    Org 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor.
  • Description
    Org 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor, significantly increases the binding of the CB1 receptor agonist [3H]CP 55,940 with pKb of 5.67; reduces food consumption in rats, produces CB1-independent hypophagic effects and does not affect the discriminative stimulus effects of anandamide (AEA).
  • Synonyms
    Org-27569;Org27569
  • Pathway
    GPCR/G Protein
  • Target
    Cannabinoid Receptor
  • Recptor
    CB1
  • Research Area
    Neurological Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    868273-06-7
  • Formula Weight
    409.95
  • Molecular Formula
    C24H28ClN3O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 52.2 mg/mL
  • SMILES
    O=C(C(N1)=C(CC)C2=C1C=CC(Cl)=C2)NCCC3=CC=C(N4CCCCC4)C=C3
  • Chemical Name
    1H-Indole-2-carboxamide, 5-chloro-3-ethyl-N-[2-[4-(1-piperidinyl)phenyl]ethyl]-

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Price MR, et al. Mol Pharmacol. 2005 Nov;68(5):1484-95.
2. Erdozain AM, et al. Biochem Pharmacol. 2012 Jan 15;83(2):260-8.
3. Fay JF, et al. J Biol Chem. 2012 Sep 28;287(40):33873-82.
4. Gamage TF, et al. Behav Pharmacol. 2014 Apr;25(2):182-5.
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