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Org 27569
CAS No. 868273-06-7
Org 27569 ( Org-27569;Org27569 )
Catalog No. M16306 CAS No. 868273-06-7
Org 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 28 | In Stock |
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| 5MG | 43 | In Stock |
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| 10MG | 73 | In Stock |
|
| 25MG | 143 | In Stock |
|
| 50MG | 267 | In Stock |
|
| 100MG | 399 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameOrg 27569
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NoteResearch use only, not for human use.
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Brief DescriptionOrg 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor.
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DescriptionOrg 27569 is a potent, selective, allosteric modulator of cannabinoid CB1 receptor, significantly increases the binding of the CB1 receptor agonist [3H]CP 55,940 with pKb of 5.67; reduces food consumption in rats, produces CB1-independent hypophagic effects and does not affect the discriminative stimulus effects of anandamide (AEA).
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SynonymsOrg-27569;Org27569
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorCB1
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Research AreaNeurological Disease
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Indication——
Chemical Information
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CAS Number868273-06-7
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Formula Weight409.95
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Molecular FormulaC24H28ClN3O
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 52.2 mg/mL
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SMILESO=C(C(N1)=C(CC)C2=C1C=CC(Cl)=C2)NCCC3=CC=C(N4CCCCC4)C=C3
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Chemical Name1H-Indole-2-carboxamide, 5-chloro-3-ethyl-N-[2-[4-(1-piperidinyl)phenyl]ethyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Price MR, et al. Mol Pharmacol. 2005 Nov;68(5):1484-95.
2. Erdozain AM, et al. Biochem Pharmacol. 2012 Jan 15;83(2):260-8.
3. Fay JF, et al. J Biol Chem. 2012 Sep 28;287(40):33873-82.
4. Gamage TF, et al. Behav Pharmacol. 2014 Apr;25(2):182-5.
2. Erdozain AM, et al. Biochem Pharmacol. 2012 Jan 15;83(2):260-8.
3. Fay JF, et al. J Biol Chem. 2012 Sep 28;287(40):33873-82.
4. Gamage TF, et al. Behav Pharmacol. 2014 Apr;25(2):182-5.
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